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17 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Optimisation of LRRK2 inhibitors and assessment of functional efficacy in cell-based models of neuroinflammation.EBI
University of Sydney
Amide-based derivatives ofß-alanine hydroxamic acid as histone deacetylase inhibitors: attenuation of potency through resonance effects.EBI
University of Sydney
The many faces of the adamantyl group in drug design.EBI
University of Sydney
Pyrazolo[1,5-a]pyrimidine acetamides: 4-Phenyl alkyl ether derivatives as potent ligands for the 18 kDa translocator protein (TSPO).EBI
University of Sydney
GABA-Activated ligand gated ion channels: medicinal chemistry and molecular biology.EBI
University of Sydney
Design, synthesis, and structure-affinity relationships of regioisomeric N-benzyl alkyl ether piperazine derivatives as sigma-1 receptor ligands.EBI
University of Sydney
Oxo-bridged isomers of aza-trishomocubane sigma (sigma) receptor ligands: Synthesis, in vitro binding, and molecular modeling.EBI
University of Sydney
Purinergic P2X(7) receptor antagonists: Chemistry and fundamentals of biological screening.EBI
University of Sydney
Novel gamma-aminobutyric acid rho1 receptor antagonists; synthesis, pharmacological activity and structure-activity relationships.EBI
University of Sydney
Two new irreversible inhibitors of dihydrodipicolinate synthase: diethyl (E,E)-4-oxo-2,5-heptadienedioate and diethyl (E)-4-oxo-2-heptenedioate.EBI
University of Sydney
Semisynthetic preparation of amentoflavone: A negative modulator at GABA(A) receptors.EBI
University of Sydney
Development of an N-Acyl Amino Acid That Selectively Inhibits the Glycine Transporter 2 To Produce Analgesia in a Rat Model of Chronic Pain.EBI
University of Sydney
Synthesis and enzymic evaluation of 4-mercapto-6-oxo-1, 4-azaphosphinane-2-carboxylic acid 4-oxide as an inhibitor of mammalian dihydroorotase.EBI
University of Sydney
Structure-activity relationships and pH dependence of binding of 8-alkyl-N5-deazapterins to dihydrofolate reductase.EBI
University of Sydney
?-aminobutyric acid(C) (GABAC) selective antagonists derived from the bioisosteric modification of 4-aminocyclopent-1-enecarboxylic acid: amides and hydroxamates.EBI
University of Sydney
GABA(C) receptors as drug targets.BDB
University of Sydney
Unsaturated phosphinic analogues of gamma-aminobutyric acid as GABA(C) receptor antagonists.BDB
University of Sydney